柽柳素及其苷在自然植物中广泛分布，同时也是槲皮素的天然黄酮衍生物。其主要药理学效应包括抗氧化、抗炎、抗病毒、抗癌、心血管效应等。药物动力学研究显示，直接吸收分布与生物合成有所不同。同时，研究表明柽柳素使用安全，因其毒性较小。本文从PubMed、中国知识数据库、万方数据库等电子数据库中获取了1976年至2023年共181篇关于柽柳素的文章。基于关键词进行柽柳素搜索，剩下121篇文章。对柽柳素的转化合成、药物动力学、药理作用和结构活性关系进行了综述。版权所有© Bentham Science Publishers；如有任何疑问，请发送电子邮件至epub@benthamscience.net。

Tamarixetin and its glycosides are widely distributed in natural plants, and they are also natural flavonoid derivatives of quercetin. Its main pharmacological effects include antioxidant, anti-inflammatory, antiviral, anticancer, cardiovascular effects, etc. The pharmacokinetics showed that the distribution of direct absorption differed from that of biosynthesis. At the same time, research shows that tamarixetin is safe to use because it has little self-toxicity. In this paper, 181 articles on tamarixetin published from 1976 to 2023 are obtained from PubMed, China Knowledge Base Database, Wanfang Data, and other electronic databases. Tamarixetin is searched based on keywords, and 121 articles remain. Transformation synthesis, pharmacokinetics, pharmacological action, and structure-activity relationship of tamarixetin were reviewed.Copyright© Bentham Science Publishers; For any queries, please email at epub@benthamscience.net.